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GPCR Cell Lines and Membranes
HTS-ready stable cell lines and membranes for high throughput screening and compound profiling in multiple assay platforms.
| Stable Cell Line Catalog Numbers | |||||||
| Receptor Family | Receptor | Species | Functional Assay Cell Lines | HExTM Cell Lines | Division-Arrested Cells | Membranes | Price |
| Adenosine | A1 | human | C1427-1![]() | Yes | Yes | inquire | |
| A2A | human | C1428-1![]() | Yes | Yes | inquire | ||
| A2B | human | C1429![]() | DC1429![]() | Yes | inquire | ||
| A2B | rat | NEWCr1429![]() | Yes | Yes | inquire | ||
| A3 | human | C1430![]() | Yes | Yes | inquire | ||
| Adrenergic | alpha 1A | human | NEWC1431-1a![]() | Yes | Yes | inquire | |
| alpha 1B | human | C1432-1![]() | Yes | Yes | inquire | ||
| alpha 1D | human | NEWC1433-1![]() | Yes | Yes | inquire | ||
| alpha 2A | human | C1434-1a C1434-1![]() | Yes | MC1434-1a MC1434-1![]() | inquire | ||
| alpha 2B | human | C1435-1![]() | Yes | MC1435-1![]() | inquire | ||
| alpha 2C | human | C1436-1![]() | Yes | Yes | inquire | ||
| beta 1 | human | C1437-1![]() | Yes | Yes | inquire | ||
| beta 2 | human | C1438-1a![]() | Yes | Yes | inquire | ||
| beta 3 | human | C1439a![]() | Yes | Yes | inquire | ||
| Anaphylatoxin | C3AR1 | human | C1222![]() | Yes | Yes | inquire | |
| C5R1 | human | C1221![]() | Yes | Yes | inquire | ||
| Angiotensin | AT1 | human | NEWH1417![]() | Yes | Yes | inquire | |
| Apelin | APJ | human | NEWC1196 C1196-1![]() | DC1196-1![]() | Yes | inquire | |
| Bile Acid | GPBA | human | NEWC1361-1a C1361-1![]() | DC1361-1a![]() | MC1361-1![]() | inquire | |
| GPBA | rat | Cr1361-1![]() | Yes | Yes | inquire | ||
| GPBA | mouse | Cm1361-1![]() | DCm1361-1![]() | Yes | inquire | ||
| Bombesin | BB1 | rat | C1211-1![]() | Yes | Yes | inquire | |
| BB1 | human | C1211![]() | Yes | Yes | inquire | ||
| BB2 | human | C1215![]() | Yes | Yes | inquire | ||
| BB3 | human | C1214![]() | H1214![]() | Yes | Yes | inquire | |
| Bradykinin | B1 | human | C1198a![]() | Yes | MC1198a![]() | inquire | |
| B1 | mouse | NEWCm1198![]() | Yes | Yes | inquire | ||
| B2 | human | NEWC1199![]() | H1199![]() | Yes | MC1199![]() | inquire | |
| Calcitonin | CALCRL | human | C1232![]() | Yes | Yes | inquire | |
| CT | human | H1231![]() | Yes | Yes | inquire | ||
| Calcium-Sensing Receptor | CASR | rat | NEWHr1233![]() | Yes | Yes | inquire | |
| CASR | human | C1233![]() | C1233![]() | DC1233![]() | MC1233![]() | inquire | |
| Cannabinoid | CB1 | human | C1229-1a C1229-1 C1229![]() | Yes | MC1229-1a![]() | inquire | |
| CB2 | human | C1230-1a C1230-1![]() | Yes | MC1230-1a![]() | inquire | ||
| GPR55 | human | C1113b![]() | H1113![]() | Yes | Yes | inquire | |
| Chemokine | CCR1 | human | NEWCG1009 C1009![]() | Yes | Yes | inquire | |
| CCR10 | human | NEWCG1018-1 C1018![]() | Yes | Yes | inquire | ||
| CCR2 | human | C1010![]() | DC1010![]() | Yes | inquire | ||
| CCR3 | human | NEWCG1011 C1011![]() | Yes | Yes | inquire | ||
| CCR4 | human | NEWCG1012 C1012![]() | DC1012![]() | Yes | inquire | ||
| CCR5 | human | NEWCG1013 C1013a C1013b![]() | DC1013b![]() | MC1013a![]() | inquire | ||
| CCR6 | human | C1014a![]() | DC1014a![]() | Yes | inquire | ||
| CCR6 | mouse | Cm1014![]() | Yes | Yes | inquire | ||
| CCR7 | human | NEWCG1015 C1015![]() | DC1015![]() | Yes | inquire | ||
| CCR8 | human | NEWCG1016 C1016a C1016![]() | Yes | Yes | inquire | ||
| CCR9 | mouse | Cm1017 CGm1017![]() | DCGm1017![]() | Yes | inquire | ||
| CCR9 | human | CG1017 C1017a C1017![]() | Yes | MC1017![]() | inquire | ||
| CMKLR1 | human | C1147 CG1147![]() | Yes | Yes | inquire | ||
| CX3CR1 | human | CG1008 C1008![]() | DCG1008![]() | MC1008![]() | inquire | ||
| CXCR1 | human | CG1001 C1001a![]() | DC1001a![]() | Yes | inquire | ||
| CXCR2 | human | CG1002 C1002![]() | DC1002![]() | Yes | inquire | ||
| CXCR3 | human | CG1003 C1003![]() | DCG1003![]() | MCG1003 MC1003![]() | inquire | ||
| CXCR4 | human | NEWCG1004 C1004-1![]() | DC1004-1![]() | MC1004-1![]() | inquire | ||
| CXCR5 | human | C1005-1a C1005 C1005-1![]() | DC1005-1a![]() | Yes | inquire | ||
| CXCR6 | human | NEWCG1006 C1006-1 C1006![]() | DCG1006![]() | Yes | inquire | ||
| CXCR7/CMKOR1 | human | C1150![]() | Yes | Yes | inquire | ||
| XCR1 | human | C1007![]() | Yes | Yes | inquire | ||
| Cholecystokinin | CCK1 | human | C1038-1a C1038![]() | Yes | MC1038-1a![]() | inquire | |
| CCK2 | human | NEWH1039![]() | Yes | Yes | inquire | ||
| Citric Acid Cycle Intermediates | GPR91 | human | C1144-1![]() | DC1144-1![]() | Yes | inquire | |
| GPR99 | human | C1132-1![]() | Yes | Yes | inquire | ||
| Corticotropin-Releasing Factor | CRF1 | human | NEWCG1040 C1040![]() | Yes | Yes | inquire | |
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